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Revised (2018) Vaughan Williams classification of antiarrhythmic drugs abridged table

Revised (2018) Vaughan Williams classification of antiarrhythmic drugs abridged table
Class 0 (HCN channel blockers)
Ivabradine
Class I (voltage-gated Na+ channel blockers)
Class Ia (intermediate dissociation):
  • Quinidine, ajmaline, disopyramide, procainamide
Class Ib (rapid dissociation):
  • Lidocaine, mexilitine
Class Ic (slow dissociation):
  • Propafenone, flecainide
Class Id (selective late sodium channel current and atrial-selective peak sodium channel current):
  • Ranolazine
Class II (autonomic inhibitors and activators)
Class IIa (beta blockers):
  • Nonselective: carvedilol, propranolol, nadolol
  • Selective: atenolol, bisoprolol, betaxolol, esmolol, metoprolol
Class IIb (nonselective beta agonists):
  • Isoproterenol
Class IIc (muscarinic M2 receptor inhibitors):
  • Atropine, hyoscine, scopolamine
Class IId (muscarinic M2 receptor activators):
  • Carbachol, pilocarpine, methacholine, digoxin
Class IIe (adenosine A1 receptor activators):
  • Adenosine
Class III (K+ channel blockers and openers)
Class IIIa (voltage dependent K+ channel blockers):
  • Amiodarone, dronedarone, dofetilide, ibutilide, sotalol
Class IV (Ca++ handling modulators)
Class IVa (surface membrane Ca++ channel blockers):
  • Diltiazem, verapamil
Class V (mechanosensitive channel blockers):
No approved medications
Class VI (gap junction channel blockers)
No approved medications
Class VII (upstream target modulators)
Angiotensin converting enzyme inhibitors
Angiotensin receptor blockers
Omega-3 fatty acids
Statins
Ca: calcium; HCN: hyperpolarization-activated cyclic nucleotide-gated; K: potassium; Na: sodium.
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