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Selection of antiemetic medications

Selection of antiemetic medications
Indication Therapeutic options
Gastroenteritis Dopamine antagonists
Serotonin antagonists
Opioid-induced nausea and vomiting Serotonin antagonists
Dopamine antagonists
  • Droperidol
Migraine-related nausea and vomiting Dopamine antagonists
  • Metoclopramide with paracetamol
  • Metoclopramide
  • Prochlorperazine
Vestibular causes of nausea and vomiting Antihistamines
Anticholinergics
Dopamine antagonists
Chemotherapy-induced nausea and vomiting Serotonin antagonists
Neurokinin-1 antagonists
Corticosteroids
  • Dexamethasone
Dopamine antagonists
  • Olanzapine, haloperidol
Benzodiazepines
  • Lorazepam
Radiation-induced nausea and vomiting Serotonin antagonists
Corticosteroids
  • Dexamethasone
Dopamine antagonists
Postoperative nausea and vomiting Dopamine antagonists
Serotonin antagonists
Antihistamines
Corticosteroids
  • Dexamethasone
Neurokinin-1 antagonists
Benzodiazepines
  • Lorazepam
Adapted with permission from: Athavale A, Athavale T, Roberts DM. Antiemetic drugs: What to prescribe and when. Aust Prescr 2020; 43:49–56. https://doi.org/10.18773/austprescr.2020.011.
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