NS5A inhibitor | Genotype 1a | Genotype 3 |
Pibrentasvir | Y93* | No single position variants¶ |
Velpatasvir | Y93 | Y93H |
Ledipasvir | K24, M28, Q30, L31, Y93 | N/A |
Elbasvir | M28, Q30, L31, Y93 | N/A |
Daclatasvir | M28, Q30, L31, Y93 | A30K, Y93H |
* Results in low level resistance in vitro (<10x shift in EC50).
¶ In vitro, no single position variant results in >3x shift in EC50. Dual A30K and Y93H results in 70x shift in EC50.
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