Formulation | Time to peak serum concentration* | Comments |
Extended-release 12-hour tablet[1,2] | 3 to 7 hours after morning dose when given every 12 hours |
|
Extended-release 24-hour tablet[3,4] | 8 to 12 hours when given every 24 hours |
|
Extended-release 24-hour capsule[5,6] (United States brand name: Theo-24) | Variable and difficult to predict; it depends on both administration time and fasting status |
|
Adapted from: Weinberger, M, Hendeles, L. Theophylline in asthma. N Engl J Med 1996; 334:1380.
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